Adrenergic Receptor Inhibitors

α adrenergic receptor

β adrenergic receptor

Adrenergic Receptor Ligands, Inhibitors, Agonists, Antagonists, Activators & Modulators

Product Name	α adrenergic receptor	β adrenergic receptor	Purity
Isoprenaline hydrochloride		β adrenergic receptor	99.86%
Norepinephrine	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.61%
Propranolol hydrochloride		β adrenergic receptor	99.96%
Propranolol		β adrenergic receptor	99.91%
Phenylephrine	α adrenergic receptor		99.98%
LM-189 free base		β2 adrenoceptor	99.45%
Zenidolol hydrochloride		β adrenergic receptor	99.74%
CL 316243		β adrenergic receptor	99.98%
D-Mannitol		Beta-3 adrenergic receptor	99.93%
Norepinephrine hydrochloride	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.95%
Phenylephrine hydrochloride	α adrenergic receptor		99.99%
Metoprolol		β1 adrenoceptor	99.97%
Atenolol		Beta-1 adrenergic receptor, Ki: 697 nM	98.85%
Clozapine	α2-adrenergic receptor, Ki: 51 nM (Inhibitor)		99.84%
Dexmedetomidine	α2-adrenergic receptor, Ki: 1.08 nM		99.93%
Dexmedetomidine hydrochloride	α2-adrenergic receptor, IC₅₀: 1.08 nM		99.94%
Prazosin hydrochloride	α adrenergic receptor		99.51%
Salbutamol		β adrenergic receptor	99.53%
Nadolol		β adrenergic receptor	99.94%
Norepinephrine bitartrate monohydrate	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.96%
(S)-Timolol maleate		β adrenergic receptor	99.80%
Mirabegron		β adrenergic receptor	99.90%
Salmeterol		β2 adrenoceptor, pEC₅₀: 9.6 β1 adrenoceptor, pEC₅₀: 6.1 β3 adrenoceptor, pEC₅₀: 5.9	99.69%
Phenylacetylglycine		β2 adrenoceptor	99.63%
Dobutamine hydrochloride	α adrenergic receptor	β adrenergic receptor	99.60%
Labetalol	α1-adrenergic receptor	β-adrenoceptor	99.94%
SR59230A		β adrenergic receptor	98.0%
Phentolamine	α adrenergic receptor		99.94%
Atipamezole	α adrenergic receptor		99.84%
Guanfacine hydrochloride	α adrenergic receptor		99.93%
L748337		Beta-3 adrenergic receptor, Ki: 4 nM Beta-2 adrenergic receptor, Ki: 204 nM Beta-1 adrenergic receptor, Ki: 390 nM	99.0%
Vilanterol trifenatate		β adrenergic receptor	99.82%
Tamsulosin	α1-adrenergic receptor		99.80%
Atipamezole hydrochloride	α adrenergic receptor		99.97%
Terazosin hydrochloride	α adrenergic receptor		99.90%
Octopamine hydrochloride	α2-adrenergic receptor		99.90%
Clonidine hydrochloride	α adrenergic receptor		99.94%
Brimonidine tartrate	α adrenergic receptor		99.68%
Acebutolol hydrochloride		β1 adrenoceptor	99.63%
Mirtazapine	α2-adrenergic receptor, pKi: 6.95		99.94%
Paliperidone	α adrenergic receptor		99.43%
Bisoprolol hemifumarate		Beta-1 adrenergic receptor	99.84%
Metoprolol succinate		β1 adrenoceptor	99.56%
Bufuralol		β-adrenoceptor	99.25%
Medetomidine hydrochloride	α2-adrenergic receptor, Ki: 1.08 nM α1-adrenergic receptor, Ki: 1750 nM		99.80%
Olodaterol		β2 adrenoceptor, EC₅₀: 0.1 nM	98.69%
Fenoterol		β adrenergic receptor	99.08%
Blonanserin	α2-adrenergic receptor, Ki: 530 (Rat c nM α1-adrenergic receptor, Ki: 26.7 (Rat nM		99.62%
Terbutaline		Beta-2 adrenergic receptor	99.77%
SR59230A hydrochloride		β adrenergic receptor	99.81%
Higenamine		β adrenergic receptor	98.91%
Indacaterol maleate		β adrenergic receptor	99.82%
Indacaterol		β adrenergic receptor	99.98%
Vibegron		β3 adrenoceptor, EC₅₀: 1.1 nM	98.03%
Methyldopa	α adrenergic receptor		98.25%
Metoprolol tartrate		β1 adrenoceptor	99.98%
Phentolamine mesylate	α adrenergic receptor		99.90%
Reboxetine mesylate	α adrenergic receptor		99.71%
Doxazosin mesylate	α adrenergic receptor		98.49%
Ecopipam hydrochloride	Alpha-2A adrenergic receptor, Ki: 731 nM		99.46%
Carazolol		β1 adrenoceptor β2 adrenoceptor β3 adrenoceptor	99.71%
DL-Norepinephrine hydrochloride	α adrenergic receptor	β adrenergic receptor	99.59%
Fenoterol hydrobromide		β adrenergic receptor	99.97%
Harmane	α2-adrenergic receptor, IC₅₀: 18 μM		99.91%
(R)-Carvedilol		β adrenergic receptor	98.78%
Vilanterol		β adrenergic receptor	99.30%
Nefazodone hydrochloride	α1-adrenergic receptor		99.94%
Piribedil	α adrenergic receptor		99.92%
Brimonidine	α adrenergic receptor		99.99%
Butaxamine hydrochloride		Beta-2 adrenergic receptor	99.87%
Talipexole dihydrochloride	α2-adrenergic receptor, IC₅₀: 25 nM		99.80%
(S)-(-)-Propranolol hydrochloride		β adrenergic receptor	99.97%
Synephrine		β adrenergic receptor	98.0%
Tamsulosin hydrochloride	α1-adrenergic receptor		99.81%
Naftopidil	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2 nM		98.14%
Terbutaline sulfate		β adrenergic receptor	99.95%
Terazosin hydrochloride dihydrate	α adrenergic receptor		99.93%
Bufuralol hydrochloride		β adrenergic receptor	≥99.0%
Bisoprolol		Beta-1 adrenergic receptor	99.78%
Pronethalol		β adrenergic receptor	99.88%
JP1302 dihydrochloride	human α2C-adrenoceptor, Ki: 28±2 nM human α2B-adrenoceptor, Ki: 1470±130 nM human α2A-adrenoceptor, Ki: 3150±50 nM rodent α2D-adrenoceptor, Ki: 1700±200 nM		99.94%
BMY 7378	rat α_1A-adrenergic receptor, Ki: 800 nM hamster alpha_1B-adrenergic receptor, Ki: 600 nM rat alpha_1D-adrenergic receptor, Ki: 2 nM		99.92%
Nicergoline	α adrenergic receptor		99.31%
Salbutamol hemisulfate		β adrenergic receptor	98.0%
Salmeterol xinafoate		β2 adrenoceptor, pEC₅₀: 9.6 β1 adrenoceptor, pEC₅₀: 6.1 β3 adrenoceptor, pEC₅₀: 5.9	99.92%
Isoetharine mesylate		β adrenergic receptor	99.05%
A-61603	α1A-adrenergic receptor		99.0%
LY 344864	rat α1-adrenergic receptor, Ki: 5.06 μM rat α2-adrenergic receptor, Ki: 3.69 μM		98.59%
Oxprenolol hydrochloride		β-adrenoceptor, Ki: 7.1 nM	99.86%
Norepinephrine tartrate	α1-adrenergic receptor α2-adrenergic receptor	Beta-1 adrenergic receptor	99.96%
Lubabegron		β adrenergic receptor	98.40%
CGP 20712 A		β adrenergic receptor	99.0%
Metaproterenol hemisulfate		β adrenergic receptor	99.86%
Asenapine	Alpha-2A adrenergic receptor, pKi: 8.9 Alpha-2C adrenergic receptor, pKi: 8.9 α1-adrenergic receptor, pKi: 8.9 Alpha-2B adrenergic receptor, pKi: 9.5		99.62%
Penbutolol sulfate		β adrenergic receptor	98.72%
(R)-Propranolol hydrochloride		β adrenergic receptor	99.36%
Esmolol hydrochloride		β-adrenoceptor	99.92%
Olodaterol hydrochloride		β2 adrenoceptor, EC₅₀: .1 nM	99.70%
Medetomidine	α2-adrenergic receptor, Ki: 1.08 nM α1-adrenergic receptor, Ki: 1750 nM		99.99%
Idazoxan hydrochloride	α adrenergic receptor		99.32%
Midodrine hydrochloride	α adrenergic receptor		99.0%
Ajmalicine	α1-adrenergic receptor α2-adrenergic receptor		99.39%
Tasipimidine sulfate	human α2A-adrenoceptor, pEC₅₀: 7.57 rat α2-adrenergic receptor, EC₅₀: 5.7 nM		99.32%
Zotepine	α adrenergic receptor		99.85%
Levobunolol hydrochloride		β adrenergic receptor	99.95%
Tulobuterol		β adrenergic receptor	99.69%
Methyldopa hydrate	α adrenergic receptor		99.95%
Etilefrine hydrochloride	α1-adrenergic receptor	Beta-1 adrenergic receptor	99.90%
Alfuzosin	α adrenergic receptor		99.86%
Ritodrine hydrochloride		β adrenergic receptor	99.82%
NP10679	Alpha-1A adrenergic receptor, IC₅₀: 0.154 μM Alpha-1A adrenergic receptor, Ki: 0.603 μM Alpha-1B adrenergic receptor, Ki: 1.92 μM Alpha-1D adrenergic receptor, Ki: 0.495 μM Alpha-2C adrenergic receptor, Ki: 3.09 μM		98.40%
Indoramin	α adrenergic receptor		99.80%
Denopamine		β adrenergic receptor	98.29%
Tizanidine	α adrenergic receptor		99.58%
Guanfacine	α adrenergic receptor		99.85%
Xamoterol hemifumarate		β adrenergic receptor	99.92%
Vatinoxan hydrochloride	α adrenergic receptor		99.79%
Levalbuterol hydrochloride		β adrenergic receptor	99.93%
BMS-466442	α adrenergic receptor, IC₅₀: ≥10 μM		98.99%
Bevantolol hydrochloride	α adrenergic receptor	β adrenergic receptor	98.98%
Clozapine (Standard)	α2-adrenergic receptor
Metoprolol-d₇ hydrochloride		β adrenergic receptor	99.71%
Talinolol		Beta-1 adrenergic receptor	99.64%
Tizanidine hydrochloride	α adrenergic receptor		99.93%
Landiolol hydrochloride		Beta-1 adrenergic receptor	99.96%
Desglymidodrine	α1A-adrenergic receptor, pKi: 5.89 α1B-adrenergic receptor, pKi: 5.16 rat alpha_1D-adrenergic receptor, pKi: 5.78 human α2A-adrenoceptor, pKi: 5.83
Efaroxan hydrochloride	α adrenergic receptor		99.94%
BRL 37344 sodium		β adrenergic receptor	99.90%
Setiptiline	α adrenergic receptor		98.03%
Atenolol (Standard)		Beta-1 adrenergic receptor
Xylometazoline hydrochloride	Alpha-1A adrenergic receptor, Ki: 0.05 μM Alpha-1B adrenergic receptor, Ki: 0.30 μM Alpha-1D adrenergic receptor, Ki: 0.15 μM Alpha-2A adrenergic receptor, Ki: 0.88 μM Alpha-2B adrenergic receptor, Ki: 1.7 μM Alpha-2C adrenergic receptor, Ki: 0.19 μM		99.94%
Metipranolol		β1 adrenoceptor, pA2: 8.3 β2 adrenoceptor, pA2: 8.4	98.36%
ARC 239 dihydrochloride	Alpha-2B adrenergic receptor		99.57%
Clorprenaline hydrochloride		β adrenergic receptor	99.90%
Spiroxatrine	α2-adrenergic receptor		99.18%
Dapiprazole hydrochloride	α1-adrenergic receptor		99.26%
Practolol		β adrenergic receptor	99.80%
Dopexamine hydrochloride		β adrenergic receptor	99.71%
Midodrine	α adrenergic receptor		99.67%
(R)-(+)-Atenolol		β adrenergic receptor	≥99.0%
Reproterol		β2 adrenoceptor
Zinterol hydrochloride		β adrenergic receptor	99.51%
Synephrine hydrochloride		β adrenergic receptor	99.66%
Detomidine hydrochloride	α adrenergic receptor		99.83%
Urapidil hydrochloride	α1-adrenergic receptor, pIC₅₀: 6.13 α2-adrenergic receptor, pIC₅₀: 4.38		99.97%
Apraclonidine hydrochloride	α adrenergic receptor		98.96%
CGP 12177 hydrochloride	α1-adrenergic receptor	Beta-1 adrenergic receptor Beta-2 adrenergic receptor Beta-3 adrenergic receptor	99.69%
Salmeterol-d₃		β adrenergic receptor	98.91%
Arformoterol tartrate		Beta-2 adrenergic receptor, Kd: 2.9 nM	99.63%
Ro 363 hydrochloride		β adrenergic receptor
BODIPY FL prazosin	α1A-adrenergic receptor, Ki: 14.5 nM α1B-adrenergic receptor, Ki: 43.3 nM		99.71%
Melperone	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM		99.84%
Celiprolol hydrochloride		β adrenergic receptor, Ki: 0.14-8.3 μM	98.93%
Amibegron hydrochloride		β adrenergic receptor	≥99.0%
Cyanopindolol		β3 adrenoceptor	99.24%
Clenproperol		β adrenergic receptor	99.44%
Buflomedil hydrochloride	rat α_1A-adrenergic receptor, Ki: 4.06 μM α1B-adrenergic receptor, Ki: 6.84 μM		99.81%
(+)-Penbutolol		β adrenergic receptor
Nifenalol hydrochloride		β-adrenoceptor	99.93%
Ulimorelin	α adrenergic receptor
Methyldopate	α adrenergic receptor		98.01%
Mabuterol		Beta-2 adrenergic receptor	99.96%
Ecopipam	Alpha-2A adrenergic receptor, Ki: 731 nM		99.77%
Abanoquil	α1-adrenergic receptor		98.07%
Dicentrine	α adrenergic receptor		99.94%
Hexoprenaline		β-adrenoceptor
HOKU-81		Beta-2 adrenergic receptor
MT-1207	α1D-adrenergic receptor, IC₅₀: 0.086 nM α1D-adrenergic receptor, Ki: 0.69 nM α1B-adrenergic receptor, IC₅₀: 0.15 nM α1B-adrenergic receptor, Ki: 1.40 nM α1A-adrenergic receptor, IC₅₀: 0.1 nM		99.96%
ORM-10921 free base	Alpha-2C adrenergic receptor, Ki: 1.4 nM		98.08%
Mibenratide		Beta-1 adrenergic receptor	99.77%
Alfuzosin hydrochloride	α adrenergic receptor		99.82%
Amidephrine	α1-adrenergic receptor
Propranolol-d₇ hydrochloride		β adrenergic receptor	98.47%
ST91	α2-adrenergic receptor		99.75%
Butyryltimolol		β adrenergic receptor	98.0%
DL 071IT		β adrenergic receptor	98.81%
Mirtazapine (Standard)	α2-adrenergic receptor
Carpipramine	α1-adrenergic receptor α2-adrenergic receptor
Etoperidone	α1-adrenergic receptor, Kd: 38 nM α2-adrenergic receptor, Kd: 570 nM
Cimaterol		β-adrenoceptor	99.13%
(RS)-Butyryltimolol		β adrenergic receptor	98.0%
Terbutaline sulfate (Standard)		β adrenergic receptor
BMY-14802 hydrochloride	α1-adrenergic receptor		98.02%
LM-189		β2 adrenoceptor
Solabegron		β adrenergic receptor	99.89%
Arformoterol		Beta-2 adrenergic receptor, Kd: 2.9 nM	99.96%
MK-761 free base		Beta-2 adrenergic receptor	99.56%
Mapenterol hydrochloride		β adrenergic receptor	99.56%
Terazosin	α adrenergic receptor
Ecopipam hydrobromide	Alpha-2A adrenergic receptor, Ki: 731 nM		99.0%
Dobutamine	α adrenergic receptor	β adrenergic receptor
Brombuterol-d₉		β adrenergic receptor	99.0%
Nadolol-d₉		β adrenergic receptor
Clorprenaline		β adrenergic receptor	99.33%
RS-79948-197	rat α2A receptor, Kd: 0.42 nM rat α2B recepter, Kd: 0.18 nM rat α2C recepter, Kd: 0.19 nM human α2A-adrenoceptor, Kd: 0.6 nM human α2B-adrenoceptor, Kd: 0.46 nM human α2C-adrenoceptor, Kd: 0.77 nM
Bunazosin	α1-adrenergic receptor		98.52%
4-Hydroxypropranolol hydrochloride		β adrenergic receptor
Fluparoxan	α2-adrenergic receptor		99.66%
Metaterol		β adrenergic receptor
Amosulalol	α1-adrenergic receptor	Beta-1 adrenergic receptor	98.69%
JP1302	human α2C-adrenoceptor, Ki: 28±2 nM human α2B-adrenoceptor, Ki: 1470±130 nM human α2A-adrenoceptor, Ki: 3150±50 nM rodent α2D-adrenoceptor, Ki: 1700±200 nM		98.68%
BMY 14802	α1-adrenergic receptor		98.96%
p-F-HHSiD hydrochloride	α1-adrenergic receptor		99.0%
α1A-AR Degrader 9c	α1A-adrenergic receptor, DC₅₀: 2.86 μM
(+)-Sotalol		β-adrenoceptor	99.89%
Bupranolol		β-adrenoceptor	98.90%
Undecylenoyl phenylalanine		β-adrenoceptor
(S)-Terazosin	α adrenergic receptor		99.90%
Xamoterol		β adrenergic receptor
α2A-AR agonist 1	Alpha-2A adrenergic receptor, EC₅₀: 0.23 nM Alpha-1A adrenergic receptor, EC₅₀: 2.5 nM Alpha-2B adrenergic receptor, EC₅₀: 16.3 nM Alpha-2C adrenergic receptor, EC₅₀: 21.3 nM		99.92%
L-771688	α adrenergic receptor		99.46%
ARC 239	human α2C-adrenoceptor, pKi: 6.95 Alpha-2C adrenergic receptor, pKi: 7.06		99.71%
Midaglizole hydrochloride	α adrenergic receptor		99.67%
Zinterol		β adrenergic receptor
Prenalterol		β1 adrenoceptor	99.18%
ST1936	α2-adrenergic receptor, Ki: 300 nM (rat) α2-adrenergic receptor, Ki: 300 nM (human) α1-adrenergic receptor, Ki: 390 nM (rat)		99.70%
Oxyfedrine		β-adrenoceptor
AGN 192836	α adrenergic receptor		99.49%
(Rac)-Rotigotine hydrochloride	Alpha-2B adrenergic receptor		98.11%
Harmane hydrochloride	α2-adrenergic receptor, IC₅₀: 18 μM
Xylometazoline	Alpha-1A adrenergic receptor, Ki: 0.05 μM Alpha-1B adrenergic receptor, Ki: 0.30 μM Alpha-1D adrenergic receptor, Ki: 0.15 μM Alpha-2A adrenergic receptor, Ki: 0.88 μM Alpha-2B adrenergic receptor, Ki: 1.7 μM Alpha-2C adrenergic receptor, Ki: 0.19 μM
Isoetharine		β adrenergic receptor
Timolol hemihydrate		β adrenergic receptor
Blonanserin dihydrochloride	α2-adrenergic receptor, Ki: 530 nM α1-adrenergic receptor, Ki: 26.7 nM
Timolol		β adrenergic receptor
(R,R)-Reboxetine mesylate	α adrenergic receptor
Sotalol		β-adrenoceptor
Dobutamine tartrate	α adrenergic receptor	β adrenergic receptor
Mivazerol	α2-adrenergic receptor
Ritodrine		β adrenergic receptor
CAXII-IN-3		Beta-2 adrenergic receptor Beta-1 adrenergic receptor Beta-3 adrenergic receptor
Etoperidone hydrochloride	α1-adrenergic receptor, Kd: 38 nM α2-adrenergic receptor, Kd: 570 nM
Metoprolol fumarate		β1 adrenoceptor
Isamoltan hydrochloride		β-adrenoceptor, IC₅₀: 8.4 nM
Bopindolol fumarate		β1 adrenoceptor β2 adrenoceptor β3 adrenoceptor
Trimazosin	α1-adrenergic receptor
Naftopidil dihydrochloride	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2
Flestolol sulfate		β adrenergic receptor
2-(2-Methoxyphenoxy)ethylamine hydrochloride	α1-adrenergic receptor		≥98.0%
Rezatomidine	α2-adrenergic receptor
Prazobind	Alpha-1A adrenergic receptor, IC₅₀: 1 nM Alpha-1B adrenergic receptor, IC₅₀: 1 nM
Nipradolol	α1-adrenergic receptor
Piribedil dihydrochloride	α adrenergic receptor
Celiprolol		β adrenergic receptor, Ki: 0.14-8.3 μM
Metoprolol-d₆ tartrate		β adrenergic receptor
ent-Levobunolol hydrochloride		β adrenergic receptor
Zolertine hydrochloride	α1B-adrenergic receptor, pKi: 6.81 (in rat liver membrane) α1A-adrenergic receptor, pKi: 6.35 (in rabbit liver membrane)
SB-206606		Beta-3 adrenergic receptor
α2AR agonist 1	α2-adrenergic receptor
Oxprenolol		β-adrenoceptor, Ki: 7.1 nM
Iloperidone carboxylic acid	human α2C-adrenoceptor, pKi: 7.32 human α2A-adrenoceptor, pKi: 6.42 rat α1-adrenergic receptor, pKi: 7.67 human α2B-adrenoceptor, pKi: 7.08
Bopindolol		β2 adrenoceptor Beta-1 adrenergic receptor Beta-3 adrenergic receptor
Nifenalol		Beta-1 adrenergic receptor
Melperone hydrochloride	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM
Fipamezole	human α2A-adrenoceptor, Ki: 9.2 nM human α2B-adrenoceptor, Ki: 17 nM human α2C-adrenoceptor, Ki: 55 nM
(E)-Guanabenz	α adrenergic receptor
α2C adrenoceptor agonist 1	Alpha-2C adrenergic receptor, EC₅₀: 108 nM Alpha-2C adrenergic receptor, Ki: 12 nM
hERG-IN-3	α1A-adrenergic receptor, IC₅₀: 270 nM	Beta-2 adrenergic receptor, IC₅₀: 14 nM
Rec 15/2615 hydrochloride	α1A-adrenergic receptor, Ki: 1.9 nM α1B-adrenergic receptor, Ki: 0.3 nM Alpha-1D adrenergic receptor, Ki: 2.6 nM
Fenoterol hydrobromide (Standard)		β adrenergic receptor
Acebutolol-d₇		β adrenergic receptor
Isamoltane hemifumarate		β-adrenoceptor, IC₅₀: 8.4 nM
Isoprenaline hemisulfate		β adrenergic receptor
S(-)-Bisoprolol fumarate		β adrenergic receptor
Butaxamine		β2 adrenoceptor
LAS190792		β2 adrenoceptor, pIC₅₀: 9.1 β3 adrenoceptor, pIC₅₀: 5.6 β1 adrenoceptor, pIC₅₀: 7.5
Ajmalicine hydrochloride	α1-adrenergic receptor α2-adrenergic receptor
S(-)-Bisoprolol		β adrenergic receptor
SM-2470	α adrenergic receptor
Acebutolol		β1 adrenoceptor
Bisoprolol fumarate		Beta-1 adrenergic receptor
Procaterol		β2 adrenoceptor
β2AR/M3-receptor agonist-1		β2 adrenoceptor, pEC₅₀: >9.2
(±)-Desisopropylpropranolol		β adrenergic receptor
(±)-Penbutolol		Beta-1 adrenergic receptor
RWJ52353	Alpha-2D adrenergic receptor, Ki: 1.5 nM Alpha-2A adrenergic receptor, Ki: 254 nM α1-adrenergic receptor, Ki: 443 nM Alpha-2B adrenergic receptor, Ki: 621 nM
Naftopidil hydrochloride	Alpha-1A adrenergic receptor, Ki: 3.7 nM Alpha-1B adrenergic receptor, Ki: 20 nM Alpha-1D adrenergic receptor, Ki: 1.2 nM
Harmane (Standard)	α2-adrenergic receptor
Ro 70‐0004	Alpha-1A adrenergic receptor, pKi: 8.9
Diacetolol-d₇		β adrenergic receptor
VUF26034		Beta-2 adrenergic receptor
Meluadrine		β2 adrenoceptor
Nemazoline	α1-adrenergic receptor α2-adrenergic receptor
ST1936 oxalate	α2-adrenergic receptor, Ki: 300 nM (rat) α2-adrenergic receptor, Ki: 300 nM (human) α1-adrenergic receptor, Ki: 390 nM (rat)
Meluadrine tartrate		β2 adrenoceptor
Cimbuterol-d₉		β adrenergic receptor
Salbutamol adipate		β adrenergic receptor
SUN-1334H free base	Alpha-1D adrenergic receptor, IC₅₀: 7.76 μM
Dapiprazole	α1-adrenergic receptor
Apraclonidine	α adrenergic receptor
Etilefrine hydrochloride (Standard)	α1-adrenergic receptor	Beta-1 adrenergic receptor
CACPD2011a-0001278239		Beta-2 adrenergic receptor
Phenylethanolamine A-d₃		β adrenergic receptor
Moprolol		Beta-1 adrenergic receptor
Pronethalol hydrochloride		β adrenergic receptor
N-5984		β-adrenoceptor
Asenapine citrate	Alpha-2A adrenergic receptor, pKi: 8.9 Alpha-2C adrenergic receptor, pKi: 8.9 α1-adrenergic receptor, pKi: 8.9 Alpha-2B adrenergic receptor, pKi: 9.5
Delequamine hydrochloride	α2-adrenergic receptor, pKi: 9.5 α1-adrenergic receptor, pKi: 5.3
Metaproterenol		β adrenergic receptor
Levalbuterol		β adrenergic receptor
Clenproperol-d₇		β adrenergic receptor
(±)-Penbutolol-d₉ hydrochloride		β adrenergic receptor
L-665871		β adrenergic receptor
Sibenadet		β2 adrenoceptor
Levobunolol		β adrenergic receptor
2-MPMDQ	α1-adrenergic receptor, Ki: 0.37 nM α2-adrenergic receptor, Ki: 1740 nM
Sulfinalol		β-adrenoceptor
Mabuterol-d₉		β adrenergic receptor
Pafenolol		Beta-1 adrenergic receptor
Agroclavine	α1-adrenergic receptor
Landiolol		Beta-1 adrenergic receptor
Clozapine dihydrochloride	α2-adrenergic receptor, Ki: 51 nM
Bunitrolol		β-adrenoceptor
SAR-150640		β3 adrenoceptor
Buflomedil	rat α_1A-adrenergic receptor, Ki: 4.06 μM α1B-adrenergic receptor, Ki: 6.84 μM
Methyldopate hydrochloride	α adrenergic receptor
AVN-101 hydrochloride	Alpha-1D adrenergic receptor, Ki: 30.2 nM Alpha-1B adrenergic receptor, Ki: 9.4 nM Alpha-2A adrenergic receptor, Ki: 1.77 nM Alpha-2C adrenergic receptor, Ki: 3.55 nM Alpha-1A adrenergic receptor, Ki: 18.9 nM Alpha-2B adrenergic receptor, Ki: 0.41 nM		99.59%
LY 344864 hydrochloride	rat α1-adrenergic receptor, Ki: 5.06 μM rat α2-adrenergic receptor, Ki: 3.69 μM
AH 11110A	α1B-adrenergic receptor
Platelet aggregation-IN-3	α2-adrenergic receptor
Ractopamine		pig β₁AR, Kd: ~25 nM pig β₂AR, Kd: ~25 nM
β2AR agonist /M-receptor antagonist-1		Beta-2 adrenergic receptor
Brombuterol-d₉ hydrochloride		β adrenergic receptor
CHF-6550		β2 adrenoceptor, pKi: 10.6
Arrestin-3 modulator-1		Beta-2 adrenergic receptor
Tasipimidine	human α2A-adrenoceptor, pEC₅₀: 7.57 rat α2-adrenergic receptor, EC₅₀: 5.7 nM
Metrenperone	α1-adrenergic receptor α2-adrenergic receptor
Zilpaterol-d₇		β adrenergic receptor
Bevantolol		Beta-1 adrenergic receptor
Doxazosin-d₈	α adrenergic receptor
Clozapine hydrochloride	α2-adrenergic receptor, Ki: 51 nM
Photoazolol-1		β-adrenoceptor
TAAR1 agonist 3	Alpha-2A adrenergic receptor, pEC₅₀: 6
Levobetaxolol		β1 adrenoceptor, IC₅₀: 33.2 nM β2 adrenoceptor, IC₅₀: 2970 nM β3 adrenoceptor, IC₅₀: 709 nM
Todralazine		β adrenergic receptor
CL 316243 free acid		β3 adrenoceptor	99.37%
Arformoterol maleate		Beta-2 adrenergic receptor, Kd: 2.9 nM
A 80426 mesylate	α2-adrenergic receptor
Levalbuterol tartrate		β adrenergic receptor
Landiolol hydrochloride (Standard)		Beta-1 adrenergic receptor
Indacaterol xinafoate		β2 adrenoceptor
Mabuterol hydrochloride		Beta-2 adrenergic receptor
Fiduxosin hydrochloride	α1A-adrenergic receptor, IC₅₀: 0.16 nM α1B-adrenergic receptor, IC₅₀: 24.9 nM α1D-adrenergic receptor, IC₅₀: 0.92 nM
Bunitrolol hydrochloride		β-adrenoceptor
PF-9404C		β adrenergic receptor
Melperone (Standard)	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM
Sulfinalol hydrochloride		β-adrenoceptor
Melperone-d₄ hydrochloride	α2-adrenergic receptor, Kd: 150 nM α1-adrenergic receptor, Kd: 180 nM		99.84%
SB251023		Beta-3 adrenergic receptor
Protokylol hydrochloride		Beta-2 adrenergic receptor
Methyldopa hydrochloride	α adrenergic receptor
Cafedrine-theodrenaline		β-adrenoceptor
4-Hydroxypropranolol-d₇ hydrochloride		β adrenergic receptor
CHIR-2279	α1-adrenergic receptor, Ki: 5 nM
RU 52583	α2-adrenergic receptor
Org 6906	α2-adrenergic receptor, pKi: 6.5
Carbuterol hydrochloride		Beta-2 adrenergic receptor
Clorprenaline-d₇		β adrenergic receptor
R 47 243	α2-adrenergic receptor
Esmolol		β adrenergic receptor
L-748328		β3 adrenoceptor, Ki: 3.7 nM
(rac)-Nebivolol-d₄		β adrenergic receptor
Cicloprolol hydrochloride		β adrenergic receptor
Pargolol hydrochloride		β adrenergic receptor
TD-5471 hydrochloride		β adrenergic receptor
OPC-28326	α adrenergic receptor
Ko-3290		β adrenergic receptor
Delequamine	α2-adrenergic receptor, pKi: 9.5 α1-adrenergic receptor, pKi: 5.3
L-770644		Beta-3 adrenergic receptor, EC₅₀: 13 nM
Azepexole dihydrochloride	α adrenergic receptor
Buflomedil hydrochloride (Standard)	rat α_1A-adrenergic receptor, Ki: 4.06 μM α1B-adrenergic receptor, Ki: 6.84 μM
Ridazolol		Beta-1 adrenergic receptor
Trimazosin hydrochloride hydrate	α1-adrenergic receptor
QF0301B	α adrenergic receptor
α1 adrenoceptor-MO-1	α adrenergic receptor
Epanolol		β adrenergic receptor
Benzquinamide	α adrenergic receptor
Fenmetozole Tosylate	α adrenergic receptor
AR-08	α adrenergic receptor

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